| 摘要 |
<p>Substituted enaminothio compounds (I) are new, where (I) excludes 4-{[(6-chloropyrid-3-yl)methyl](methyl)amino}furan-2(5H)-thione, 4-{[(6-chloropyrid-3-yl)methyl]amino}furan-2(5H)-thione, 4-{[(6-chloropyrid-3-yl)methyl](methyl)amino}thiophen-2(5H)-thione and 4-{[(6-chloropyrid-3-yl)methyl](ethyl)amino}thiophen-2(5H)-thione. Substituted enaminothio compounds of formula (I) are new, where (I) excludes 4-{[(6-chloropyrid-3-yl)methyl](methyl)amino}furan-2(5H)-thione, 4-{[(6-chloropyrid-3-yl)methyl]amino}furan-2(5H)-thione, 4-{[(6-chloropyrid-3-yl)methyl](methyl)amino}thiophen-2(5H)-thione and 4-{[(6-chloropyrid-3-yl)methyl](ethyl)amino}thiophen-2(5H)-thione. A : pyrid-2-yl, pyrid-4-yl or pyrid-3-yl (all optionally substituted in 6th-position by F, Cl, Br, CH 3, CF 3or CF 3O), pyridazin-3-yl (optionally substituted in 6-position by Cl or CH 3), or pyrazin-3-yl, 2-chloropyrazin-5-yl or 1,3-thiazol-5-yl (all optionally substituted in 2nd-position by Cl or CH 3), or pyrimidinyl, pyrazolyl, thiophenyl, oxazolyl, isoxazolyl, 1,2,4-oxadiazolyl, isothiazolyl, 1,2,4-triazolyl or 1,2,5-thiadiazolyl (all optionally substituted by F, Cl, Br, CN, NO 2, 1-4C-alkyl (optionally substituted by F and/or Cl), 1-3C-alkylthio (optionally substituted by F and/or Cl), or 1-3C-alkylsulfonyl (optionally substituted by F and/or Cl), or 1-3C-alkylsulfonyl (optionally substituted by F and/or Cl)), or pyridine group of formula (a); X : halo, alkyl or haloalkyl; Y 1>halo, alkyl, haloalkyl, haloalkoxy, azido or CN; B 1>O, S or methylene; R 1>H, alkyl, haloalkyl, alkenyl, haloalkenyl, alkynyl, cycloalkyl, cyclodialkyl, halocycloalkyl, alkoxy or halocyclodialkyl; R 2>H or halo; and R 3>H or alkyl. [Image] [Image] ACTIVITY : Pesticide; Arthropodicide; Insecticide; Arachnicide; Nematocide; Acaricide; Fungicide; Antibacterial; Virucide; Herbicide; Antimicrobial; Antifouling. MECHANISM OF ACTION : None given.</p> |
