发明名称 INDOLE DERIVATIVE OR PHARMACEUTICALLY ACCEPTABLE SALT THEREOF
摘要 <p>PROBLEM TO BE SOLVED: To provide a compound having EPreceptor antagonism, a pharmaceutically acceptable salt thereof, a pharmaceutical composition containing the same and a medical use thereof.SOLUTION: There is provided a compound having EPreceptor antagonism and represented by the general formula (I), where A is a pyridine ring or the like, Yis a Calkylene group or the like, Yis a single bond or the like, Ris a hydrogen atom or the like, Ris a Ccycloalkylene group with a ring substituted by a Calkyl group or the like, Ris a carboxyl group or the like, Ris a hydrogen atom, Ris a hydrogen atom or the like, Ris a Calkyl group or the like and Rrepresents a hydrogen atom or the like, or a pharmaceutically acceptable salt thereof. The compound (I) can further used as a therapeutic agent or prophylactic agent for various symptoms of LUTS, especially OABs.</p>
申请公布号 JP2015137266(A) 申请公布日期 2015.07.30
申请号 JP20140010730 申请日期 2014.01.23
申请人 KISSEI PHARMACEUTICAL CO LTD;KYORIN PHARMACEUTICAL CO LTD 发明人 TAYA KAZUYA;KONDO ATSUSHI;KONDO TATSUHIRO;KAWAMURA NAOHIRO;SETO SHIGEKI
分类号 C07D401/12;A61K31/4439;A61K31/506;A61P13/02;A61P43/00;C07D401/06;C07D401/14;C07D405/14;C07D491/056 主分类号 C07D401/12
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