发明名称 Fungicidal 4-substituted-3-{phenyl[(heterocyclylmethoxy)imino]methyl}-1,2,4-oxadizol-5(4H)-one derivatives
摘要 The present invention provides fungicidal 4-substituted-3-{phenyl[(heterocyclylmethoxy)imino]methyl}-1,2,4-oxadiazol-5(4H)-one derivatives of formula (I); wherein A represents a pyridyl or thiazole group and X1, Y1 to Y5 represent independently different substituents.
申请公布号 US9090600(B2) 申请公布日期 2015.07.28
申请号 US201214344579 申请日期 2012.09.10
申请人 BAYER INTELLECTUAL PROPERTY GMBH 发明人 Braun Christoph;Sawada Haruko;Lachaise Helene;Brunet Stephane;Rinolfi Philippe;Dubost Christophe;Coqueron Pierre-Yves;Maechling Simon;Rebstock Anne-Sophie;Wachendorff-Neumann Ulrike
分类号 A01N43/836;C07D417/12;C07D417/14;C07D413/12;C07D413/14;C07D277/40;C07D271/07;C07D213/75;C07D213/73;C07D213/74;C07D277/46;C07D277/48;A01N43/82;C07D231/16;C07D231/38;A01N55/00;C07F7/10;C07F7/08 主分类号 A01N43/836
代理机构 Ostrolenk Faber LLP 代理人 Ostrolenk Faber LLP
主权项 1. A compound of formula (I) wherein X1 is selected from the group consisting of a hydrogen atom, a formyl group, substituted or non-substituted C1-C8-alkyl, substituted or non-substituted C3-C8-cycloalkyl, a substituted or non-substituted C2-C8-alkenyl, substituted or non-substituted C2-C8-alkynyl, and a substituted or non-substituted C1-C8-alkylcarbonyl;A is selected from A1 or A2: wherein Z1 is selected from the group consisting of a hydrogen atom, a halogen atom, a nitro group, an amino group, an hydroxyamino group, an hydroxy group, a cyano group, substituted or non-substituted C1-C8-alkoxyamino group, substituted or non-substituted C1-C8-alkylamino, substituted or non-substituted C2-C8-alkenylamino, substituted or non-substituted C2-C8-alkynylamino, substituted or non-substituted C3-C10-cycloalkylamino, substituted or non-substituted C3-C10-cycloalkenylamino, substituted or non-substituted C5-C12-fused bicycloalkylamino, substituted or non-substituted C5-C12-fused bicycloalkenylamino, substituted or non-substituted di-C1-C8-alkylamino, substituted or non-substituted phenylamino, substituted or non-substituted heterocyclylamino, and a group of formula QC(=U)NRa wherein:Q is selected from the group consisting of a hydrogen atom, substituted or non-substituted C1-C8-alkyl, substituted or non-substituted C3-C8-cycloalkyl, substituted or non-substituted C2-C8-alkenyl, substituted or non-substituted C3-C8-cycloalkenyl, substituted or non-substituted C2-C8-alkynyl, substituted or non-substituted C1-C8-alkoxy, substituted or non-substituted C2-C8-alkenyloxy, substituted or non-substituted C2-C8-alkynyloxy, substituted or non-substituted C1-C8-alkylamino, substituted or non-substituted C1-C8-alkylsulfenyl, substituted or non-substituted C2-C8-alkenylsulfenyl, substituted or non-substituted C2-C8-alkynylsulfenyl, substituted or non-substituted arylsulfenyl, substituted or non-substituted aryl, substituted or non-substituted heterocyclyl, substituted or non-substituted C5-C12-fused bicycloalkyl, substituted or non-substituted C5-C12-fused bicycloalkenyl, substituted or non-substituted C5-C12-benzofused carbocyclyl, substituted or non-substituted C5-C12-benzofused heterocyclyl, substituted or non-substituted cycloalkoxy; substituted or non-substituted cycloalkenyloxy, substituted or non-substituted aryloxy; substituted or non-substituted heterocyclyloxy, substituted or non-substituted C5-C12-fused bicycloalkoxy, substituted or non-substituted C5-C12-fused bicycloalkenyloxy, substituted or non-substituted C5-C12-benzofused carbocyclyloxy, and substituted or non-substituted C5-C12-benzofused heterocyclyloxy;U is an oxygen atom or a sulfur atom;Ra is selected from the group consisting of a hydrogen atom, a hydroxy group, substituted or non-substituted C1-C8-alkyl, substituted or non-substituted C3-C8-cycloalkyl, substituted or non-substituted C2-C8-alkenyl, substituted or non-substituted C2-C8-alkynyl, substituted or non-substituted C1-C8-alkoxy, substituted or non-substituted C3-C10-cycloalkenyl, substituted or non-substituted C5-C12-fused bicycloalkyl, substituted or non-substituted C5-C12-fused bicycloalkenyl, substituted or non-substituted aryl, substituted or non-substituted heterocyclyl, substituted or non-substituted C1-C8-alkylcarbonyl, substituted or non-substituted aryloxycarbonyl, and substituted or non-substituted C1-C8-alkoxycarbonyl;Z2, Z3 and Z4 independently are selected from the group consisting of a hydrogen atom, a halogen atom, substituted or non-substituted C1-C8-alkyl, substituted or non-substituted C3-C8-cycloalkyl, C2-C8-alkenyl, substituted or non-substituted C2-C8-alkynyl, and substituted or non-substituted C1-C8-alkoxy;Y1 to Y5 independently are selected from the group consisting of a hydrogen atom, a halogen atom, a nitro group, a cyano group, substituted or non-substituted carbaldehyde O—(C1-C8-alkyl)oxime, a pentafluoro-λ6-sulfenyl group, substituted or non-substituted C1-C8-alkyl, substituted or non-substituted C3-C8-cycloalkyl, substituted or non-substituted C1-C8-halogenoalkyl having 1 to 5 halogen atoms, C2-C8-alkenyl, substituted or non-substituted C2-C8-alkynyl, substituted or non-substituted C1-C8-alkoxy, substituted or non-substituted C1-C8-halogenoalkoxy having 1 to 5 halogen atoms, substituted or non-substituted C1-C8-alkylsulfenyl, substituted or non-substituted C2-C8-alkenyloxy, substituted or non-substituted C3-C8-alkynyloxy, substituted or non-substituted N—(C1-C8-alkoxy)-C1-C8-alkanimidoyl, substituted or non-substituted N—(C1-C8-alkoxy)-C1-C8-halogenoalkanimidoyl having 1 to 5 halogen atoms, substituted or non-substituted C1-C8-alkoxycarbonyl, substituted or non-substituted C1-C8-alkylcarbonyloxy, substituted or non-substituted C1-C8-alkylsulfinyl, substituted or non-substituted C1-C8-alkylsulfonyl, substituted or non-substituted phenoxy, substituted or non-substituted phenylsulfenyl, substituted or non-substituted aryl, substituted or non-substituted tri(C1-C8-alkyl)-silyloxy, substituted or non-substituted tri(C1-C8-alkyl)-silyl, substituted or non-substituted heterocyclyl, and substituted or non-substituted heterocyclyloxy; salts, N-oxides, metallic complexes and metalloidic complexes thereof or (E) and (Z) isomers and mixtures thereof.
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