| 主权项 |
1. Compounds of the formula (I) in which R1 denotes Y or —(CY2)n—Ar, R2 denotes Y, —(CY2)p—(C[YR6])n—R7 or -alk-R7, R3 denotes Y or CN, R4 denotes Y, Hal, —(CY2)p—COOY or —(CY2)p—CO—NYY, R5 denotes A, Hal, —(CY2)p—OY, —(CY2)p—NYY, —(CY2)p—COOY, —(CY2)p—CO—NYY or —(CY2)p—NY—COY, R6 denotes Y, Hal, —(CY2)n—NYY, —(CY2)n—NY—COO—(CY2)n—SiA3, —(CY2)n—COOY, —CO—NYY, —CO—NY—(CY2)n—OY, —CO—NY—(CY2)n—NYY or SO2A, R7 denotes —(CY2)p—Ar or —(CY2)p-Het1, X denotes CH2, O, S or a single bond, Y denotes H or A, A denotes unbranched or branched alkyl having 1, 2, 3, 4, 5, 6, 7, 8, 9 or 10 C atoms, where 1, 2, 3, 4, 5, 6 or 7 H atoms may be replaced, independently of one another, by Hal, Alk denotes alkenyl having 1, 2, 3, 4, 5 or 6 C atoms, where 1, 2, 3 or 4 H atoms may be replaced, independently of one another, by Hal and/or OY, Ar denotes phenyl which is unsubstituted or mono-, di- or trisubstituted by Hal, A, CN, —(CY2)p—OY, —(CY2)p—NYY, —(CY2)p—COOY, —(CY2)p—CO—NYY or —(CY2)p—NY—COY, Het1 denotes mono- or bicyclic heteroaryl having 2, 3, 4, 5, 6, 7, 8 or 9 C atoms and 1, 2, 3 or 4 N, O and/or S atoms, which may be unsubstituted or mono-, di- or trisubstituted by Hal, A, CN, —(CY2)p—OY, —(CY2)p—NYY, —(CY2)p—COOY, —(CY2)p—CO—NYY, —(CY2)p—NY—COY or —SO2-Het2, Het2 denotes a monocyclic saturated heterocycle having 2, 3, 4, 5, 6 or 7 C atoms and 1, 2, 3 or 4 N, O and/or S atoms, which may be unsubstituted or monosubstituted by A, Hal denotes F, Cl, Br or I, m denotes 0, 1, 2, 3 or 4, and n, p, s, independently of one another, denote 0, 1, 2, 3, 4, 5 or 6, and/or physiologically acceptable salts, tautomers and/or stereoisomers thereof, including mixtures thereof in all ratios. |
