发明名称 HYDROXY FORMAMIDE DERIVATIVES AND THEIR USE
摘要 Disclosed are compounds having the formula (I): wherein R1, R2 and R3 are as defined herein, and methods of making and using the same, including use as inhibitors of BMP1, TLL1 and/or TLL2 and in treatment of diseases associated with BMP1, TLL1 and/or TLL2 activity.
申请公布号 CA2936467(A1) 申请公布日期 2015.07.16
申请号 CA20152936467 申请日期 2015.01.09
申请人 GLAXOSMITHKLINE INTELLECTUAL PROPERTY (NO.2) LIMITED 发明人 DOWDELL, SARAH E.;EIDAM, HILARY SCHENCK;ELBAN, MARK;FOX, RYAN MICHAEL;HAMMOND, MARLYS;HILFIKER, MARK A.;HOANG, TRAM H.;KALLANDER, LARA S.;LAWHORN, BRIAN GRIFFIN;MANNS, SHARADA;PHILP, JOANNE;WASHBURN, DAVID G.;YE, GUOSEN
分类号 C07D407/04;A61K31/431;A61P43/00;C07D307/24;C07D307/68 主分类号 C07D407/04
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