发明名称 A CRYSTALLINE MONOHYDRATE OF THE COMPOUND OF FORMULA (IV) AND A PROCESS FOR PREPARING THE SAME
摘要 <p>The invention relates to processes for preparing compounds having the formula (I) and crystalline forms thereof, wherein Ar is aryl or heteroaryl, L is an optional alkylene linker, and R2, R3, R4, and R5, are as defined in the specification herein, which compounds are useful as kinase inhibitors, in particular, inhibitors of protein tyrosine kinase and p38 kinase.</p>
申请公布号 IN6567DEN2014(A) 申请公布日期 2015.07.10
申请号 IN2014DE06567 申请日期 2014.08.05
申请人 BRISTOL-MYERS SQUIBB HOLDINGS IRELAND 发明人 CHEN BANG-CHI;DROGHINI ROBERTO;LAJEUNESSE JEAN;DIMARCO JOHN D.;GALELLA MICHAEL;CHIDAMBARAM RAMAKRISHNAN
分类号 C07D471/04;C07C235/28;C07C237/42;C07D277/56;C07D417/12;C07D417/14;C07D463/00 主分类号 C07D471/04
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