发明名称 |
Vannfrie aripiprazol-krystaller F, fremgangsmåte for fremstilling derav samt farmasøytisk preparat |
摘要 |
<p>The present invention provides low-hygroscopic forms of aripiprazole and processes for the preparation thereof which will not convert to a hydrate or lose their original solubility even when a medicinal preparation containing the aripiprazole anhydride crystals is stored for an extended period.</p> |
申请公布号 |
NO336262(B1) |
申请公布日期 |
2015.07.06 |
申请号 |
NO20080001632 |
申请日期 |
2008.04.02 |
申请人 |
OTSUKA PHARMACEUTICAL CO., LTD. |
发明人 |
TOMINAGA MICHIAKI;BANDO TAKUJI;AOKI SATOSHI;KAWASAKI JUNICHI;ISHIGAMI MAKOTO;TANIGUCHI YOUICHI;YABUUCHI TSUYOSHI;FUJIMOTO KIYOSHI;NISHIOKA YOSHIHIRO;KOBAYASHI NORIYUKI;FUJIMURA TSUTOMO;TAKAHASHI MASANORI;ABE KAORU;NAKAGAWA TOMONORI;SHINHAMA KOICHI;UTSUMI NAOTO;OI YOSHIHIRO;YAMADA SHOHEI;TOMIKAWA KENJI |
分类号 |
C07D215/22;A61K;A61K9/14;A61K9/16;A61K9/20;A61K31/4704;A61K31/496;A61K31/501;A61P;A61P1/08;A61P3/04;A61P15/10;A61P25/00;A61P25/04;A61P25/16;A61P25/18;A61P25/22;A61P25/28;A61P25/32;B01D9/02;C07D;C07D215/227 |
主分类号 |
C07D215/22 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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