发明名称 METHOD FOR PRODUCING 5-HYDROXYPIPERIDINE-2-CARBOXYLIC ACID
摘要 A method for producing (2S,5S)/(2R,5R)-5-hydroxypiperidine-2-carboxylic acid indicated by formula (10), the method being characterized in including a step for removing protection from hydroxyl groups in a compound represented by formula (7) and synthesizing a compound represented by formula (8). (In the formula, P indicates a protecting group; R3 indicates an alkyl group having 1-4 carbon atoms; and A indicates an alkyl group having 1-10 carbon atoms, an aryl group having 6-12 carbon atoms, an alkyloxy group having 1-4 carbon atoms, or an aralkyloxy group having 7-20 carbon atoms.) (In the formula, R3 indicates an alkyl group having 1-4 carbon atoms; and A indicates an alkyl group having 1-10 carbon atoms, an aryl group having 6-12 carbon atoms, an alkyloxy group having 1-4 carbon atoms, or an aralkyloxy group having 7-20 carbon atoms.)
申请公布号 WO2015099126(A1) 申请公布日期 2015.07.02
申请号 WO2014JP84518 申请日期 2014.12.26
申请人 API CORPORATION 发明人 TAKEHARA, JUN;MURAI, MASATO;OHTANI, TAKASHI;MAEDA, TOMOKO;HIDAKA, TSUGIHIKO
分类号 C07D211/60;C07B61/00;C07C233/47;C07C309/66;C07D498/08 主分类号 C07D211/60
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