发明名称 SERINE/THREONINE KINASE INHIBITORS FOR THE TREATMENT OF HYPERPROLIFERATIVE!DISEASES
摘要 Compounds having the formula I wherein R2, X and Z as defined herein are inhibitors of ERK kinase. Also disclosed are compositions and methods for treating hyperproliferative disorders.
申请公布号 EP2888247(A1) 申请公布日期 2015.07.01
申请号 EP20130759395 申请日期 2013.08.27
申请人 ARRAY BIOPHARMA, INC.;GENENTECH, INC. 发明人 BLAKE, JIM;CHEN, HUIFEN;CHICARELLI, MARK;GAUDINO, JOHN;GAZZARD, LEWIS;KINTZ, SAM;MOHR, PETE;ROBARGE, KIRK;SCHWARZ, JACOB;ZHOU, AIHE
分类号 C07D401/14;A61K31/4375;A61K31/472;A61K31/4725;A61P35/00;C07D217/22;C07D401/12;C07D471/04 主分类号 C07D401/14
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