发明名称 4-(8-methoxy-1-((1-methoxypropan-2-yl)-2-(tetrahydro-2H-pyran-4-yl)-1 H-imidazo[4,5-C]quinolin-7-yl)-3,5-dimethylisoxazole and its use as bromodomain inhibitor
摘要 Novel quinoline compounds pharmaceutical compositions containing such compounds and their use in therapy.
申请公布号 US9067936(B2) 申请公布日期 2015.06.30
申请号 US201214237905 申请日期 2012.08.15
申请人 GlaxoSmithKline LLC 发明人 Demont Emmanuel Hubert;Jones Katherine Louise;Watson Robert J.
分类号 C07D471/00;A61K31/44;C07D471/04;A61K31/4745 主分类号 C07D471/00
代理机构 代理人 Brink Robert H.
主权项 1. A compound of formula (I) which is 4-(8-methoxy-1-(1-methoxypropan-2-yl)-2-(tetrahydro-2H-pyran-4-yl)-1H-imidazo[4,5-c]quinolin-7-yl)-3,5-dimethylisoxazoleor a salt thereof.
地址 Wilmington DE US