发明名称 |
6-ALKENYL AND 6-PHENYLALKYL SUBSTITUTED 2-QUINOLINONES AND 2-QUINOXALINONES AS POLY (ADP-RIBOSE) POLYMERASE INHIBITORS |
摘要 |
<p>THE PRESENT INVENTION PROVIDES COMPOUNDS OF FORMULA (I) AND COMPOUNDS OF FORMULA (VII-A) AS WELL AS PHARMACEUTICAL COMPOSITIONS COMPRISING SAID COMPOUNDS AND THEIR USE AS PARP INHIBITORS WHEREIN N,R1,R2,R3,R4,R5,R6,R7,RE,RD AND X HAVE DEFINED MEANINGS.</p> |
申请公布号 |
MY154363(A) |
申请公布日期 |
2015.06.15 |
申请号 |
MY2004PI04774 |
申请日期 |
2004.11.18 |
申请人 |
JANSSEN PHARMACEUTICA N.V. |
发明人 |
MABIRE, DOMINIQUE JEAN-PIERRE;GUILLEMONT, JÉRÔME EMILE GEORGES;VAN DUN, JACOBUS ALPHONSUS;SOMERS, MARIA VICTORIA FRANCISCA;WOUTERS, WALTER BOUDEWIJN |
分类号 |
C07D215/227;C07D215/22;C07D241/44;C07D401/06;C07D401/14;C07D403/06;C07D405/06;C07D405/14;C07D407/06;C07D409/12 |
主分类号 |
C07D215/227 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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