发明名称 |
CRYSTALLINE FORM OF (S)-(2-(6-CHLORO-7-METHYL-1H-BENZO[D]IMIDAZOL-2-YL)-2-METHYLPYRROLIDIN-1 -YL)(5-METHOXY-2-(2H-1,2,3-TRIAZOL-2-YL)PHENYL)METHANONE AND ITS USE AS OREXIN RECEPTOR ANTAGONISTS |
摘要 |
The invention relates to crystalline forms of (S)-(2-(6-chloro-7-methyl-1H-benzo[d]imidazol-2- yl)-2-methylpyrrolidin-1-yl)(5-methoxy-2-(2H-1,2,3-triazol-2-yl)phenyl)methanone, processes for the preparation thereof, pharmaceutical compositions containing such crystalline forms, pharmaceutical compositions prepared from such crystalline forms, and their use as a medicament, especially as orexin receptor antagonists. |
申请公布号 |
WO2015083070(A1) |
申请公布日期 |
2015.06.11 |
申请号 |
WO2014IB66508 |
申请日期 |
2014.12.02 |
申请人 |
ACTELION PHARMACEUTICALS LTD |
发明人 |
BOSS, CHRISTOPH;BROTSCHI, CHRISTINE;GUDE, MARKUS;HEIDMANN, BIBIA;SIFFERLEN, THIERRY;VON RAUMER, MARKUS;WILLIAMS, JODI, T. |
分类号 |
C07D403/14;A61K31/4192;A61P25/00 |
主分类号 |
C07D403/14 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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