发明名称 CRYSTALLINE FORMS OF N-(TERT-BUTOXYCARBONYL)-3-METHYL-L-VALYL-(4R)-4-((7-CHLORO-4-METHOXY-1-ISOQUINOLINYL)OXY)-N-((1R,2S)-1-((CYCLOPROPYLSULFONYL)CARBAMOYL)-2-VINYLCYCLOPROPYL)-L-PROLINAMIDE
摘要 The present disclosure generally relates to crystalline forms of N-(tert-butoxycarbonyl)-3-methyl-L-valyl-(4R)-4-((7-chloro-4-methoxy-1-isoquinolinyl)oxy)-N-((1R,2S)-1-((cyclopropylsulfonyl)carbamoyl)-2-vinylcyclopropyl)-L-prolinamide. The present disclosure also generally relates to a pharmaceutical composition comprising one or more of the crystalline forms, as well as methods of using the crystalline forms in the treatment of Hepatitis C virus (HCV) and methods for obtaining such crystalline forms.
申请公布号 HRP20150458(T1) 申请公布日期 2015.06.05
申请号 HR2015P000458T 申请日期 2015.04.28
申请人 BRISTOL-MYERS SQUIBB HOLDINGS IRELAND 发明人 PERRONE, ROBERT KEVIN;WANG, CHENCHI;YING, WILLIAM;SONG, ANNE I.
分类号 C07D401/12;A61K31/44;A61P31/14 主分类号 C07D401/12
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