发明名称 |
BICYCLIC HETEROCYCLES AS BET PROTEIN INHIBITORS |
摘要 |
<p>The present invention relates to bicyclic heterocycles which are inhibitors of BET proteins such as BRD2, BRD3, BRD4, and BRD-t and are useful in the treatment of diseases such as cancer.</p> |
申请公布号 |
WO2015081246(A1) |
申请公布日期 |
2015.06.04 |
申请号 |
WO2014US67691 |
申请日期 |
2014.11.26 |
申请人 |
INCYTE CORPORATION |
发明人 |
YUE, EDDY W.;COMBS, ANDREW P. |
分类号 |
C07D471/04;A61K31/437;A61P9/00;A61P29/00;A61P31/12;A61P35/00 |
主分类号 |
C07D471/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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