| 发明名称 |
PROCESS FOR PREPARING AN INTERMEDIATE TO MU OPIOID RECEPTOR ANTAGONISTS |
| 摘要 |
<p>The invention provides an efficient method for preparing 3-endo-(S-azabicyclo[3.2.1]oct-3-yl)benzamide by hydrogenation, under controlled conditions, of an amino-protected 3-(8-azabicyclo[3.2.1]oct-2-en-3-yl)benzamide intermediate in which the amino-protecting group is removable by catalytic hydrogenation.</p> |
| 申请公布号 |
CA2690606(C) |
申请公布日期 |
2015.05.26 |
| 申请号 |
CA20082690606 |
申请日期 |
2008.07.15 |
| 申请人 |
THERAVANCE, INC. |
发明人 |
COLSON, PIERRE-JEAN;YU, YING;LONG, DANIEL D.;STERGIADES, IOANNA |
| 分类号 |
C07D451/02 |
主分类号 |
C07D451/02 |
| 代理机构 |
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