发明名称 PYRAZOLE DERIVATIVE AND USE THEREOF FOR MEDICAL PURPOSES
摘要 The present invention provides pyrazole derivatives, uses thereof for medical purposes and so on. More particularly, the present invention relates to pharmaceuticals useful for the prevention or treatment of constipation, which comprise as an active ingredient 3-(3-{4-[3-(β-D-glucopyranosyloxy)-5-isopropyl-1H-pyrazol-4-ylmethyl]-3-methylphenoxy}propylamino)-2,2-dimethylpropionamide, or a pharmaceutically acceptable salt thereof. The pharmaceuticals of the present invention exert an effect of increasing the frequency of bowel movement or the like, and are useful for the prevention or treatment of constipation.
申请公布号 US2015141631(A1) 申请公布日期 2015.05.21
申请号 US201314399093 申请日期 2013.05.02
申请人 Kissei Pharmaceutical Co., Ltd. 发明人 Isaji Masayuki;Takemura Masaaki;Isawa Hidetoshi;Hotei Yukihiko;Miyashita Itaru
分类号 C07H17/02 主分类号 C07H17/02
代理机构 代理人
主权项 1. A pharmaceutical for use in the prevention or treatment of constipation, which comprises as an active ingredient 3-(3-{4-[3-(β-D-glucopyranosyloxy)-5-isopropyl-1H-pyrazol-4-ylmethyl]-3-methylphenoxy}propylamino)-2,2-dimethylpropionamide, or a pharmaceutically acceptable salt thereof.
地址 Matsumoto-shi, Nagano JP