发明名称 |
PROCESS FOR THE SYNTHESIS OF AN INDOLEAMINE 2,3-DIOXYGENASE INHIBITOR |
摘要 |
<p>The present application is directed to processes and intermediates for making 4-({2-[(aminosulfonyl)amino]ethyl}amino)-N-(3-bromo-4-fluorophenyl)-N'-hydroxy-1,2,5-oxadiazole-3-carboximidamide, which is an inhibitor of indoleamine 2,3-dioxygenase, useful in the treatment of cancer and other disorders.</p> |
申请公布号 |
WO2015070007(A1) |
申请公布日期 |
2015.05.14 |
申请号 |
WO2014US64531 |
申请日期 |
2014.11.07 |
申请人 |
INCYTE CORPORATION |
发明人 |
TAO, MING;FRIETZE, WILLIAM;MELONI, DAVID J.;WENG, LINGKAI;ZHOU, JIACHENG;PAN, YONGCHUN |
分类号 |
C07D271/08;A61K31/4245;A61P35/00;C07D413/04 |
主分类号 |
C07D271/08 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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