发明名称 HETEROBICYCLOARYL RORC2 INHIBITORS AND METHODS OF USE THEREOF
摘要 The present invention provides compounds, pharmaceutical compositions, methods of inhibiting RORy activity and/or reducing the amount of IL-17 in a subject, and methods of treating various medical disorders using such compounds and pharmaceutical compositions.
申请公布号 WO2015015378(A3) 申请公布日期 2015.05.14
申请号 WO2014IB63383 申请日期 2014.07.24
申请人 PFIZER INC. 发明人 BLINN, JAMES, ROBERT;FLICK, ANDREW, CHRISTOPHER;WENNERSTÅL, GÖRAN, MATTIAS;JONES, PETER;KAILA, NEELU;KIEFER, JAMES, RICHARD, JR.;KURUMBAIL, RAVI, G.;MENTE, SCOT, RICHARD;MEYERS, MARVIN, JAY;SCHNUTE, MARK, EDWARD;THORARENSEN, ATLI;XING, LI;ZAMARATSKI, EDOUARD;ZAPF, CHRISTOPH, WOLFGANG
分类号 C07D401/14;A61K31/454;A61K31/497;A61K31/506;A61K31/519;A61K31/5355;A61P29/02;A61P37/08;C07D401/04;C07D407/14;C07D413/04;C07D413/14;C07D417/14;C07D471/04;C07D487/04 主分类号 C07D401/14
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