发明名称 |
PHOSPHATIDYL INOSITOL 3-KINASE INHIBITOR AND APPLICATION METHOD THEREOF |
摘要 |
<p>PROBLEM TO BE SOLVED: To provide a small molecule inhibitor of phosphatidyl inositol 3-kinase (PI3K) relating to many malignant diseases such as ovarian cancer, cervical cancer, breast cancer, colon cancer, rectal cancer and glioblastoma.SOLUTION: There is provided a quinoxaline sulfonamide compound represented by the formula (I).</p> |
申请公布号 |
JP2015091860(A) |
申请公布日期 |
2015.05.14 |
申请号 |
JP20150003368 |
申请日期 |
2015.01.09 |
申请人 |
EXELIXIS INC |
发明人 |
BAJJALIEH WILLIAM;BANNEN LYNNE CANNE;BROWN S DAVID;KEARNEY PATRICK;MAC MORRISON B;MARLOWE CHARLES K;NUSS JOHN M;TESFAI ZEROM;WANG YONG;XU WEI |
分类号 |
C07D241/44;A61K31/498;A61K31/4985;A61K31/501;A61K31/506;A61K31/5377;A61K31/551;A61K31/63;A61P35/00;A61P35/02;C07D401/12;C07D401/14;C07D403/12;C07D403/14;C07D405/12;C07D405/14;C07D409/12;C07D413/12;C07D417/12;C07D471/04 |
主分类号 |
C07D241/44 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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