发明名称 NOVEL INDANESULFAMIDE DERIVATIVE.
摘要 <p>A novel indanesulfamide compound, such as N-[(1S)-2,2,5,7-tetrafluoro-2,3-dihydro-1H-inden-1-yl]- sulfamide, N-[(1S)-2,2,4,7-tetrafluoro-2,3-dihydro-1H- inden-1-yl]sulfamide and (+)-N-(2,2,4,6,7- pentafluoro-2,3-dihydro-1H-inden-1-yl)sulfamide, or a pharmaceutically acceptable salt thereof has an effect of improving the severity (score) of an attack in a mouse kindling model and therefore can be expected to serve as a therapeutic agent for epilepsy.</p>
申请公布号 MX2014015492(A) 申请公布日期 2015.05.08
申请号 MX20140015492 申请日期 2013.06.17
申请人 EISAI R&D MANAGEMENT CO., LTD. 发明人 YUJI KAZUTA;TORU WATANABE;KEIICHI SORIMACHI;MINAKO SAITO;YOICHI KITA;TOSHIAKI TANAKA;HIROYUKI HIGASHIYAMA;TAKAHISA HANADA;TETSUYUKI TERAMOTO;TAKASHI KOSASA;YUKIO ISHIKAWA
分类号 C07C307/08;A61K31/18;A61K31/277;A61P25/08 主分类号 C07C307/08
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