发明名称 ANDROGEN RECEPTOR MODULATING COMPOUNDS
摘要 Compounds of formula (I)wherein Rto R, A, B and E are as defined in the claims and pharmaceutically acceptable salts and esters thereof, are disclosed. The compounds of formula (I) possess utility as tissue-selective androgen receptor modulators (SARM) and are particularly useful as medicaments in the treatment of prostate cancer and other AR dependent conditions and diseases where AR antagonism is desired.
申请公布号 EA021170(B1) 申请公布日期 2015.04.30
申请号 EA20120070597 申请日期 2010.10.27
申请人 ORION CORPORATION 发明人 WOHLFAHRT GERD;TOERMAEKANGAS OLLI;SALO HARRI;HOEGLUND IISA;KARJALAINEN ARJA;KNUUTTILA PIA;HOLM PATRIK;RASKU SIRPA;VESALAINEN ANNIINA
分类号 C07D231/14;A61K31/416;A61K31/42;A61K31/438;A61K31/44;A61K31/4523;A61K31/497;A61K31/5377;A61P35/00;C07D401/12;C07D403/12;C07D405/12;C07D413/12;C07D417/12 主分类号 C07D231/14
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