发明名称 |
TREATMENT USING BRUTON'S TYROSINE KINASE INHIBITORS AND IMMUNOTHERAPY |
摘要 |
Combinations of Bruton's tyrosine kinase (Btk) inhibitors, e.g., l-((R)-3-(4-amino-3-(4- phenoxyphenyl)- 1 H-pyrazolo [3,4-d]pyrimidin- 1 -yl)piperidin- 1 -yl)prop-2-en- 1 -one, with immunotherapy are provided. Also provided are methods of treating cancers, and autoimmune disorders by administering combinations of Bruton's tyrosine kinase (Btk) inhibitors, e.g., 1- ((R)-3-(4-amino-3-(4-phenoxyphenyl)-lH-pyrazolo[3,4-d]pyrimidin-l-yl)piperidin-l-yl)prop-2- en-l-one, and an immune checkpoint inhibitor. |
申请公布号 |
WO2015061752(A1) |
申请公布日期 |
2015.04.30 |
申请号 |
WO2014US62278 |
申请日期 |
2014.10.24 |
申请人 |
PHARMACYCLICS, INC.;THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY |
发明人 |
LEVY, RONALD;CHANG, BETTY;NG, PATRICK;SAGIV-BARFI, IDIT |
分类号 |
A61K39/395;A61K31/519;A61P35/00 |
主分类号 |
A61K39/395 |
代理机构 |
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代理人 |
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地址 |
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