发明名称 IMIDAZOLYL ANALOGS AS SYK INHIBITORS
摘要 The present invention provides novel imidazole analogs of Formula I which are potent inhibitors of spleen tyrosine kinase, and are useful in the treatment and prevention of diseases mediated by said enzyme, such as asthma, COPD, rheumatoid arthritis, and cancer.
申请公布号 EP2863913(A1) 申请公布日期 2015.04.29
申请号 EP20130807108 申请日期 2013.06.18
申请人 MERCK SHARP & DOHME CORP.;MERCK CANADA INC. 发明人 LIM, JONGWON;REUTERSHAN, MICHAEL, H.;ELLIS, JOHN MICHAEL;CHILDERS, KALEEN KONRAD;DONOFRIO, ANTHONY;ALTMAN, MICHAEL, D.;HAIDLE, ANDREW, M.;ZABIEREK, ANNA;CHRISTOPHER, MATTHEW;GRIMM, JONATHAN;BURCH, JASON;FRANCESCO, MARIA EMILIA DI;PETROCCHI, ALESSIA;BEAULIEU, CHRISTIAN;TRUONG, VOUY LINH;NORTHRUP, ALAN, B.;BLOUIN, MARC
分类号 A61K31/50;A61K31/501;C07D401/14;C07D403/12;C07D403/14 主分类号 A61K31/50
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