发明名称 |
N-(2-aminophenyl)-4-[N-(pyridine-3-yl)-methoxycarbonyl-aminomethyl]-benzamide (MS-275) polymorph B |
摘要 |
The crystalline Polymorph B of N-(2-aminophenyl)-4-[N-(pyridine-3-yl)methoxy-carbonyaminomethyl]benzamide (MS-275) of formula I;
is described, as well as the process for the production of said compound, and its use as a medicament for the treatment of selected diseases. |
申请公布号 |
USRE45499(E1) |
申请公布日期 |
2015.04.28 |
申请号 |
US201414201684 |
申请日期 |
2014.03.07 |
申请人 |
Bayer Intellectual Property GmbH |
发明人 |
Schneider Matthias;Gottfried Michael;Geisler Jens;Winter Gabriele;Suzuki Joji;Ando Tomoyuki;Honjo Masaru |
分类号 |
C07D213/56;A01N43/40;A61K31/4406 |
主分类号 |
C07D213/56 |
代理机构 |
Wilson Sonsini Goodrich & Rosati |
代理人 |
Wilson Sonsini Goodrich & Rosati |
主权项 |
1. Crystalline N-(2-aminophenyl)-4-[N-(pyridine-3-yl)methoxycarbonylamino-methyl]-benzamide polymorph B of formula Isubstantially free of N-(2-aminophenyl)-4-[N-(pyridine-3 yl)methoxy-carbonylamino-methyl]-benzamide polymorph A. |
地址 |
Monheim am Rhein DE |