发明名称 CRYSTALLINE SOLVATES OF (1S)-1,5-ANHYDRO-1-C-(3-((PHENYL) METHYL) PHENYL)- D-GLUCITOL DERIVATIVES WITH ALCOHOLS AS SGLT2 INHIBITORS FOR THE TREATMENT OF DIABETES SGLT2 (1S)-15--1-C-(3 -(()))-D-
摘要 The present invention relates to physical crystal structures of a compound of the formula I: wherein R 1 , R 2 , R 2a , R 3 and R 4 are as defined herein, especially pharmaceutical compositions containing structures of compound I or II, processes for preparing same, intermediates used in preparing same, and methods of treating diseases such as diabetes using such structures.
申请公布号 HK1127359(A1) 申请公布日期 2015.04.24
申请号 HK20090106471 申请日期 2009.07.16
申请人 ASTRAZENECA AB 发明人 JACK Z. GOUGOUTAS;HILDEGARD LOBINGER;SRIVIDYA RAMAKRISHNAN;PRASHANT P. DESHPANDE;JEFFREY T. BIEN;CHIAJEN LAI;CHENCHI WANG;PETER RIEBEL;JOHN ANTHONY GROSSO;ALEXANDRA A. NIRSCHL;JANAK SINGH;JOHN D. DIMARCO
分类号 C07H;A61K;A61P 主分类号 C07H
代理机构 代理人
主权项
地址