发明名称 TRICYCLIC TETRAHYDROQUINOLINE ANTIBACTERIAL AGENTS
摘要 Described herein are antibacterial compounds of formula I,;;methods for making the compounds, pharmaceutical compositions containing the compounds and methods of treating bacterial infections utilizing the compounds and pharmaceutical composition.
申请公布号 US2015111884(A1) 申请公布日期 2015.04.23
申请号 US201414580870 申请日期 2014.12.23
申请人 Zoetis LLC 发明人 Curtis Michael P.;Johnson Timothy Allan;Lall Manjinder S.;Toogood Peter Laurence;Warmus Joseph S.
分类号 C07D498/20;A01N47/38 主分类号 C07D498/20
代理机构 代理人
主权项 1. A compound of formula I: wherein: R1 is selected from the group consisting of: which are optionally substituted with R2; R2 is C1-6alkyl or phenyl optionally substituted with halo;X and Y are independently H, halo or C1-6 alkyl; or a salt, solvate, or a hydrate thereof; provided that when R1 is moiety (b) and R2 is phenyl, at least one of X and Y is halo.
地址 Florham Park NJ US