发明名称 |
TRICYCLIC TETRAHYDROQUINOLINE ANTIBACTERIAL AGENTS |
摘要 |
Described herein are antibacterial compounds of formula I,;;methods for making the compounds, pharmaceutical compositions containing the compounds and methods of treating bacterial infections utilizing the compounds and pharmaceutical composition. |
申请公布号 |
US2015111884(A1) |
申请公布日期 |
2015.04.23 |
申请号 |
US201414580870 |
申请日期 |
2014.12.23 |
申请人 |
Zoetis LLC |
发明人 |
Curtis Michael P.;Johnson Timothy Allan;Lall Manjinder S.;Toogood Peter Laurence;Warmus Joseph S. |
分类号 |
C07D498/20;A01N47/38 |
主分类号 |
C07D498/20 |
代理机构 |
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代理人 |
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主权项 |
1. A compound of formula I: wherein:
R1 is selected from the group consisting of: which are optionally substituted with R2;
R2 is C1-6alkyl or phenyl optionally substituted with halo;X and Y are independently H, halo or C1-6 alkyl; or a salt, solvate, or a hydrate thereof;
provided that when R1 is moiety (b) and R2 is phenyl, at least one of X and Y is halo. |
地址 |
Florham Park NJ US |