发明名称 Composto de alfa-(n-sulfonamido) acetamida como um inibidor de produção de peptídeo beta amiloide
摘要 <p>The present invention provides novel intermediates and processes for preparing them. They are useful for preparing (2R)-2-[[(4-chlorophenyl)-sulfonyl][[2-fluoro-4-(1,2,4-oxadiazol-3-yl)phenyl]methyl]amino]-5,5,5-trifluoropentanamide which is suitable for the treatment of Alzheimer's disease and other conditions associated with ²-amyloid peptide.</p>
申请公布号 BRPI0818837(A2) 申请公布日期 2015.04.22
申请号 BR2008PI18837 申请日期 2008.10.14
申请人 BRISTOL-MYERS SQUIBB COMPANY 发明人 JOHN E. STARRETT;JR.;KEVIN W. GILLMAN;RICHARD E. OLSON
分类号 C07D271/06;A61K31/4245;A61P25/28 主分类号 C07D271/06
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