发明名称 SERINE/THREONINE KINASE INHIBITORS
摘要 <p>Compounds having the formula I wherein Z, Z1 Z2 Z, R3a, R3b and Rb and as defined herein are inhibitors of ERK kinase. Also disclosed are compositions and methods for treating hyperproliferative disorders.</p>
申请公布号 EP2681215(B1) 申请公布日期 2015.04.22
申请号 EP20120709429 申请日期 2012.02.28
申请人 ARRAY BIOPHARMA, INC.;GENENTECH, INC. 发明人 BLAKE, JAMES F.;CHEN, HUIFEN;CHICARELLI, MARK JOSEPH;DEMEESE, JASON;GARREY, RUSTAM;GAUDINO, JOHN J.;KAUS, ROBERT J.;KOLAKOWSKI, GABRIELLE R.;MARLOW, ALLISON L.;MOHR, PETER J.;REN, LI;SCHWARZ, JACOB;SIEDEM, CHRISTOPHER S.;THOMAS, ALLEN A.;WALLACE, ELI;WENGLOWSKY, STEVEN MARK;BOYD, STEVEN
分类号 C07D471/04;A61K31/519;A61P35/00 主分类号 C07D471/04
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