发明名称 PROCESS FOR THE PREPARATION OF N-PROTECTED (5S)-5-(1,3-THIAZOLIDIN-3-YLCARBONYL)PYRROLIDIN-3-ONE
摘要 <p>The present invention provides a process for the preparation of an N-protected (5S)-5-(1,3-thiazolidin-3-ylcarbonyl)pyrrolidin-3-one of Formula III. The invention also provides a process for the preparation of {(2S,4S)-4-[4-(3-methyl-1-phenyl-1H-pyrazol-5- yl)piperazin-1-yl]pyrrolidin-2-yl}(1,3-thiazolidin-3-yl)methanone, or salts thereof, using the N-protected (5S)-5-(1,3-thiazolidin-3-ylcarbonyl)pyrrolidin-3-one of Formula III.</p>
申请公布号 WO2015019238(A8) 申请公布日期 2015.04.16
申请号 WO2014IB63486 申请日期 2014.07.28
申请人 RANBAXY LABORATORIES LIMITED 发明人 GIRI, PRABHAT;TENDOLKAR, ACHYUT;KAPOOR, ASHWINI, KUMAR;BARMAN, DHIREN CHANDRA;NATH, ASOK;PRASAD, MOHAN
分类号 C07D417/06;C07D417/14 主分类号 C07D417/06
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