发明名称 |
PROCESS FOR THE PREPARATION OF N-PROTECTED (5S)-5-(1,3-THIAZOLIDIN-3-YLCARBONYL)PYRROLIDIN-3-ONE |
摘要 |
<p>The present invention provides a process for the preparation of an N-protected (5S)-5-(1,3-thiazolidin-3-ylcarbonyl)pyrrolidin-3-one of Formula III. The invention also provides a process for the preparation of {(2S,4S)-4-[4-(3-methyl-1-phenyl-1H-pyrazol-5- yl)piperazin-1-yl]pyrrolidin-2-yl}(1,3-thiazolidin-3-yl)methanone, or salts thereof, using the N-protected (5S)-5-(1,3-thiazolidin-3-ylcarbonyl)pyrrolidin-3-one of Formula III.</p> |
申请公布号 |
WO2015019238(A8) |
申请公布日期 |
2015.04.16 |
申请号 |
WO2014IB63486 |
申请日期 |
2014.07.28 |
申请人 |
RANBAXY LABORATORIES LIMITED |
发明人 |
GIRI, PRABHAT;TENDOLKAR, ACHYUT;KAPOOR, ASHWINI, KUMAR;BARMAN, DHIREN CHANDRA;NATH, ASOK;PRASAD, MOHAN |
分类号 |
C07D417/06;C07D417/14 |
主分类号 |
C07D417/06 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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