发明名称 3-ARYLPYRAZOLOPYRIDINE DERIVATIVE
摘要 Provided is a compound represented by general formula (I) [where X is a hydrogen atom or a halogen atom, and R is an optionally substituted aryl group or an optionally substituted heteroaryl group], or a pharmaceutically acceptable salt thereof, which has an excellent LCAT activation effect and is useful as the active ingredient of a therapeutic agent or prophylactic agent for arteriosclerosis, arteriosclerotic heart disease, coronary heart disease (including heart failure, myocardial infarction, angina, cardiac ischemia, cardiovascular disturbance, and angioplasty-related restenosis), cerebrovascular disease (including stroke and cerebral infarction), peripheral vascular disease (including diabetic vascular complication), dyslipidemia, hypo-HDL-cholesterolemia, and kidney disease, and particularly as the active ingredient of an antiarteriosclerosis agent.
申请公布号 WO2015050148(A1) 申请公布日期 2015.04.09
申请号 WO2014JP76256 申请日期 2014.10.01
申请人 DAIICHI SANKYO COMPANY,LIMITED 发明人 KUBOTA, HIDEKI;KOBAYASHI, HIDEKI;UEDA, KIYONO;ARAI, MASAMI;NISHI, TATSUYA;TERASAKA, NAOKI
分类号 A61K31/437;A61K31/444;A61K31/4545;A61K31/5377;A61P3/06;A61P9/00;A61P9/10;A61P13/12;A61P43/00 主分类号 A61K31/437
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