Self-reactive arms and prodrugs comprising same

摘要

The present invention relates to a compound of general formula (I):;
in which:
X is OH, NH2, NHOH or RNH, where R may be a linear or branched, saturated or unsaturated, C1-C10 alkyl radical,Y is H, or an electron-withdrawing group, in particular selected from NO2, CF3 or a halogen,R1 and R2 are H or a linear or branched, saturated or unsaturated, C1-C10 alkyl radical,F is a reactive functional group that can be activated by click chemistry.

主权项

1. A compound having a general formula (I):wherein:
X is OH, NH2, NHOH or R′NH wherein R′ is a linear or branched, saturated or unsaturated, C1 to C10 alkyl radical, Y is an electron-withdrawing group, R1 and R2, independently of one another, are H or a linear or branched, saturated or unsaturated, C1 to C10 alkyl radical, F is a reactive function group activable by click chemistry.