发明名称 |
Process for preparing benzimidazole compounds comprising single step cyclisation |
摘要 |
<p>Provided are methods for the synthesis of heterocyclic compounds such as benzimidazole carboxylic acid core structures having Formula Ia-1 and their synthetic intermediates: wherein Z, X1, X2, X5, R2 and R10 are as defined herein. Compounds of Formula Ia-1 and their synthetic intermediates can be used to prepare heterocyclic derivatives such as benzimidazole derivatives.</p> |
申请公布号 |
IL188273(A) |
申请公布日期 |
2015.03.31 |
申请号 |
IL20070188273 |
申请日期 |
2007.12.19 |
申请人 |
ASTRAZENECA AB;ARRAY BIOPHARMA INC.;JOHN LEONARD;JOHN DEMATEI;SAGAR SHAKYA;MATTHEW CHARLES EVANS;JAMES GAIR FORD;ANTHONY D. PISCOPIO;BRUNO P. HACHE;SIMON MARK POINTON;KOEN PEETERS;TIMOTHY JOHN LILLEY |
发明人 |
JOHN LEONARD;JOHN DEMATEI;SAGAR SHAKYA;MATTHEW CHARLES EVANS;JAMES GAIR FORD;ANTHONY D. PISCOPIO;BRUNO P. HACHE;SIMON MARK POINTON;KOEN PEETERS;TIMOTHY JOHN LILLEY |
分类号 |
C07D |
主分类号 |
C07D |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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