发明名称 CRYSTALLINE FORM OF METHYL ((1S)-1-(((2S)-2-(5-(4'-(2-((2S)-1-((2S)-2-((METHOXYCARBONYL)AMINO)-3-METHYLBUTANOYL)-2-PYRROLIDINYL)-1H-IMIDAZOL-5-YL)-4-BIPHENYLYL)-1H-IMIDAZOL-2-YL)-1-PYRROLIDINYL)CARBONYL)-2-METHYLPROPYL)CARBAMATE DIHYDROCHLORIDE SALT
摘要 <p>The present disclosure generally relates to a crystalline form of methyl ((1S)-1-(((2S>2-(5-(4'-(2-((2S)-1-((2S)-2--((methoxycarbonyl)amino)-3-methylbutanoyl)-2-pyrrolidinyl)-1H-imidazol-5-yl)-4-biphenylyl)-1H-imidazol-2-yl)-1-pyrrolidinyl)carbonyl)-2-methylpropyl)carbamate dihydrochloride salt. The present disclosure also generally relates to a pharmaceutical composition comprising a crystalline form, as well of methods of using a crystalline form in the treatment of Hepatitis C and methods for obtaining such crystalline form.</p>
申请公布号 CA2695729(C) 申请公布日期 2015.03.31
申请号 CA20082695729 申请日期 2008.07.31
申请人 BRISTOL-MYERS SQUIBB COMPANY 发明人 KIM, SOOJIN;GAO, QI;YANG, FUKANG
分类号 C07D403/12;A61K31/4178;A61P31/12 主分类号 C07D403/12
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