发明名称 NOVEL PHTHALAZINONE-PYRROLOPYRIMIDINECARBOXAMIDE DERIVATIVES
摘要 The compounds of formula (1), in which R1, R7, R8, R9, R10, R17, R18, R19, R20 and m have the meanings as given in the description, are novel effective inhibitors of type 4 and 5 phosphodiesterase.
申请公布号 TN2013000439(A1) 申请公布日期 2015.03.30
申请号 TN20130000439 申请日期 2013.10.29
申请人 TAKEDA GMBH 发明人 STENGEL, THOMAS;MAIER, THOMAS;MANN, ALEXANDER;STADLWIESER, JOSEF;FLOCKERZI, DIETER;PAHL, ANDREAS;BENEDIKTUS, EWALD;HESSMANN, MANUELA;KANACHER, TOBIAS;HUSSONG, RAGNA;ZITT, CHRISTOF;HOLST, HANS CHRISTOF;HUMMEL, ROLF-PETER;VIERTELHAUS, MARTIN;TENOR, HERMANN;DUNKERN, TORSTEN;HATZELMANN, ARMIN;HESSLINGER, CHRISTIAN
分类号 A61K31/519;A61P11/00;C07D487/04 主分类号 A61K31/519
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