发明名称 Solid Compositions Comprising a Salt of Aminocarboxylic Acid
摘要 The present disclosure provides solid compositions comprising a stabilized salt of aminocarboxylic acid. Pharmaceutical compositions comprising [(1R,5S,6S)-6-(aminomethyl)-3-ethylbicyclo[3.2.0]hept-3-en-6-yl]acetic acid monobenzenesulfonate in combination with appropriate additives are also provided.
申请公布号 US2015079166(A1) 申请公布日期 2015.03.19
申请号 US201414553341 申请日期 2014.11.25
申请人 Daiichi Sankyo Company, Limited 发明人 Tajiri Shinichiro;Takemura Masami;Yoshinaga Shinji
分类号 A61K31/195;A61K47/12;A61K9/20;A61K47/38;A61K47/10;A61K47/26 主分类号 A61K31/195
代理机构 代理人
主权项 1. A pharmaceutical composition comprising: [(1R,5S,6S)-6-(aminomethyl)-3-ethylbicyclo[3.2.0]hept-3-en-6-yl]acetic acid monobenzenesulfonate of formula (I): (i) one or two or more components selected from the group consisting of D-mannitol, lactose, corn starch, and crystalline cellulose; and (ii) any one or both of carmellose calcium and sodium carboxymethyl starch.
地址 Tokyo JP