发明名称 RAPAMYCIN ANALOGUES AND THEIR PHARMACEUTICAL USE
摘要 Novel rapamycin analogues and methods for their production with FKBP and/or MIP inhibitory activity with reduced mTOR inhibitory activity with therapeutic potential e.g. as bacterial virulence inhibitors.
申请公布号 WO2015004455(A3) 申请公布日期 2015.03.12
申请号 WO2014GB52091 申请日期 2014.07.09
申请人 ISOMERASE THERAPEUTICS LIMITED 发明人 GREGORY, MATTHEW ALAN;KENDREW, STEVEN GARY;MOSS, STEVEN JAMES;WILKINSON, BARRIE
分类号 C07D498/18;A01N43/90;A61K31/439;A61P31/00;C12P17/18 主分类号 C07D498/18
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