发明名称 |
SUBSTITUTED PIPERIDINES AS GPR119 MODULATORS FOR THE TREATMENT OF METABOLIC DISORDERS |
摘要 |
<p>The present invention relates to compounds of general formula I, wherein R1, LP, HetAr, Ar, and n are as defined in the application, which have valuable pharmacological properties, and in particular bind to the GPR119 receptor and modulate its activity.</p> |
申请公布号 |
EP2718288(B1) |
申请公布日期 |
2015.03.11 |
申请号 |
EP20120726611 |
申请日期 |
2012.06.06 |
申请人 |
BOEHRINGER INGELHEIM INTERNATIONAL GMBH;NEUROCRINE BIOSCIENCES, INC. |
发明人 |
HECKEL, ARMIN;HIMMELSBACH, FRANK;LANGKOPF, ELKE;NOSSE, BERND;ASHWEEK, NEIL, J.;HARRIOTT, NICOLE |
分类号 |
C07D413/14;A61K31/454;A61K31/4545;A61K31/497;A61K31/506;A61P3/10;C07D401/14 |
主分类号 |
C07D413/14 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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