主权项 |
1. A pharmaceutical composition for parenteral administration of a pharmaceutical active ingredient, the composition comprising:
a) an aqueous solution or mixture; b) a pharmaceutical active ingredient; and c) a solubility enhancer comprising at least one of oleoyl-diethylenetriamine-PEG-lactobionate, oleoyl-N-(3-aminopropyl)propane-1,3-diamine-undecaethylene-glycol-methyl-ether-lactobionate, oleoy-(aminopropylamino)ethanoyl-mPEG-lactobionate, myristoyl-diethylenetriamine-dodecaethylene-glycol-lactobionate, myristoyl-triethylenetetramine-dodecaethylene-glycol-lactobionate, oleoyl-triethylenetetramine-dodecaethylene-glycol-lactobionate, and oleoyl-triethylenetetramine-pentadecaethylene-glycol-lactobionate. |