发明名称 BRANIMYCIN DERIVATIVES AND THEIR USE FOR THE TREATMENT OF BACTERIAL INFECTIOUS DISEASES
摘要 Compounds are disclosed that have a formula represented by Formula (I) wherein A, B, R1, R2 and R3 are as defined herein. Novel compounds of the invention may be prepared as a pharmaceutical composition, and may be useful in the treatment of infectious diseases, in particular bacterial infectious diseases. The compounds may be active against a specific enzyme in the bacterial DNA replicative process, DNA polymerase IIIE.
申请公布号 WO2015028095(A1) 申请公布日期 2015.03.05
申请号 WO2013EP68056 申请日期 2013.09.02
申请人 GALAPAGOS NV 发明人 DUDFIELD, PHILIP JOHN;LOWTHER, JOHN;DELACHAUME, CAROLE ANNIE JOSETTE;LÉPINE, RENAUD HENRI MARCEL;ROTH DIT BETTONI, ROMAIN VINCENT RAPHAËL;GUILLAUME, JULIE MARIE-HÉLÈNE MARTHE;THYS, AMBER PAULA MARCELLA;BARON, ANNE CATHERINE;CANOVA, SOPHIE LUCIENNE JEANNE;WITZIG, ROBERT;DOYON, JULIEN GEORGES PIERRE-OLIVIER;TOUMI, MATHIEU PAUL;HANSSKE, FRIEDRICH GEORG
分类号 C07D493/04;A61K31/343;A61P31/04 主分类号 C07D493/04
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