| 发明名称 | Prodrugs of secondary amine compounds | ||
| 摘要 | The present invention relates to compounds of Formula I:; | ||
| 申请公布号 | US8969337(B2) | 申请公布日期 | 2015.03.03 |
| 申请号 | US201213714830 | 申请日期 | 2012.12.14 |
| 申请人 | Alkermes Pharma Ireland Limited | 发明人 | Blumberg Laura Cook;Lowe John A.;Almarsson Orn;Alvarez Juan;Zeidan Tarek A. |
| 分类号 | C07D495/04;A61K47/48 | 主分类号 | C07D495/04 |
| 代理机构 | Elmore Patent Law Group, P.C. | 代理人 | Elmore Carolyn S.;Issac Roy P.;Elmore Patent Law Group, P.C. |
| 主权项 | 1. A compound selected from: wherein R1 is —C(O)OC(R4)(R5)—OC(O)(G12)mR6; R4 and R5 are from hydrogen; G12 is selected from absent, NH, CH2, —S— or —O—; m is 0 or 1; R6 is selected from C13-C26-alkyl, substituted C13-C26-alkyl, C13-C26-alkenyl, substituted C13-C26-alkenyl, C13-C26-alkynyl, substituted C13-C26-alkynyl, C13-C26-cycloalkyl, and substituted C13-C26-cycloalkyl. | ||
| 地址 | Dublin IE | ||