发明名称 |
PROCESS AND INTERMEDIATES FOR THE SYNTHESIS OF (3-ALKYL-5-PIPERIDIN-1-YL-3,3A-DIHYDRO-PYRAZOLO[1,5-A]PYRIMIDIN-7-YL)-AMINO DERIVATIVES AND INTERMEDIATES |
摘要 |
<p>This application discloses a novel process to synthesize (3-alkyl-5-piperidin-1-yl-3,3a-dihydro-pyrazolo[1,5-a]pyrimidin-7-yl)-amino derivatives, and intermediates useful in the synthesis thereof. The subject (3-alkyl-5-piperidin-1-yl-3,3a-dihydro-pyrazolo[1,5-a]pyrimidin-7-yl)-amino derivatives are useful as cyclin-dependent kinase inhibitor compounds (CDK inhibitors) in pharmaceutical preparations.</p> |
申请公布号 |
CA2661737(C) |
申请公布日期 |
2015.02.10 |
申请号 |
CA20072661737 |
申请日期 |
2007.08.17 |
申请人 |
SCHERING CORPORATION |
发明人 |
CHEN, FRANK XING;KEERTIKAR, KARTIK M.;KUO, SHEN-CHUN;LEE, HONG-CHANG;RAGHAVAN, RAMANI R.;WU, GEORGE G.;XIE, JI |
分类号 |
C07D487/04 |
主分类号 |
C07D487/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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