发明名称 PROCESS FOR THE PREPARATION OF 2-(TRIAZINYLCARBONYL)SULFONANILIDES
摘要 <p>The invention relates to a method, which is based on the oxidative ring opening of a compound with an oxindole structure, for producing substituted 2-(triazinylcarbonyl) sulfonanilides of formula (1-1) proceeding from an N-sulfonyl-substituted 3-triazinyl oxindole of formula (2-1), to the thus produced 2-(triazinylcarbonyl) sulfonanilides of formula (1-1), and to the use thereof as intermediate products for the synthesis of fine chemicals and active substances in the agricultural field. Furthermore, the invention relates to a multistage method for producing N-alkyl-N-[2-(1,3,5-triazin-2-ylcarbonyl)phenyl]alkansulfonamides of formula (4-1) proceeding from a 3-(alkylsulfanyl)-1,3-dihydro-2H-indol-2-on of formula (7-1), wherein the multistage method also has said oxidative opening as a sub-step, and to the 2-(triazinylcarbonyl) sulfonanilides of formula (1-1), said sulfonanilides being obtained by means of the oxidative ring opening and used as intermediates in the multistage method.</p>
申请公布号 EP2655346(B1) 申请公布日期 2015.01.21
申请号 EP20110807678 申请日期 2011.12.19
申请人 BAYER INTELLECTUAL PROPERTY GMBH 发明人 KARIG, GUNTER;FORD, MARK, JAMES;SIEGEL, KONRAD
分类号 C07D251/20;A01N43/66;C07D403/04 主分类号 C07D251/20
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