发明名称 |
BENZOQUINOLINE INHIBITORS OF VESICULAR MONOAMINE TRANSPORTER 2 |
摘要 |
PROBLEM TO BE SOLVED: To provide new benzoquinoline inhibitors of vesicular monoamine transporter 2 (VMAT2), pharmaceutical compositions thereof, and methods of use thereof.SOLUTION: This invention provides a compound of a structural formula I or salt thereof, where R-Rare independently selected from the group consisting of hydrogen and deuterium; and at least one of R-Ris deuterium. |
申请公布号 |
JP2015007124(A) |
申请公布日期 |
2015.01.15 |
申请号 |
JP20140185634 |
申请日期 |
2014.09.11 |
申请人 |
AUSPEX PHARMACEUTICALS INC |
发明人 |
THOMAS G GANT;MANOUCHEHR SHAHBAZ |
分类号 |
C07D455/06;A61K31/40;A61K31/4515;A61K31/454;A61K31/4745;A61K31/5415;A61K31/551;A61K31/5513;A61K31/5517;A61K31/553;A61K31/554;A61K45/00;A61P1/16;A61P25/14;A61P43/00 |
主分类号 |
C07D455/06 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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