发明名称 TRANS-4-[[(5S)-5-[[[3,5-BIS(TRIFLUOROMETHYL)PHENYL]METHYL] (2-METHYL-2H-TETRAZOL-5-YL)AMINO]-2,3,4,5-TETRAHYDRO-7,9-DIMETHYL-1H-1-BENZAZEPIN-1-YL]METHYL]-CYCLOHEXANECARBOXYLIC ACID
摘要 Abstract Compounds of a formula entitled, trans-4-[[(5S)-5-[[[3,5-bis(trifluoromethyl)phenyl]methyl] (2-methyl-2H-tetrazol- 5-yl)amino]-2,3,4,5-tetrahydro-7,9-dimethyl-1H-1-benzazepin-1-yl] methyl]- cyclohexanecarboxylic acid, as a free acid or a pharmaceutically acceptable salt thereof, hydrate, and hydrate in crystalline form; pharmaceutical formulations; and methods of use are disclosed.
申请公布号 CA2764425(C) 申请公布日期 2015.01.06
申请号 CA20102764425 申请日期 2010.06.28
申请人 ELI LILLY AND COMPANY 发明人 CHEN, XINCHAO;FRANK, SCOTT ALAN;REMICK, DAVID MICHAEL;PEDERSEN, STEVEN WAYNE
分类号 C07D403/12;A61K31/55;A61P9/10 主分类号 C07D403/12
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