发明名称 Drug Delivery Technology
摘要 The invention provides a pharmaceutical composition for the transmucosal delivery of a PDE5 inhibitor, said composition comprising a PDE5 inhibitor and a carrier in which said PDE5 inhibitor is soluble or forms a suspension or emulsion. The invention also provides a pharmaceutical composition comprising a PDE5 inhibitor for use in inhibiting PDE activity in vivo, where in said use said composition is delivered by the transmucosal route.
申请公布号 US2015005307(A1) 申请公布日期 2015.01.01
申请号 US201214367312 申请日期 2012.12.19
申请人 LondonPharma Ltd. 发明人 Sams Martin James;High Juliet Victoria;Jamieson Paul Andrew;Booles Clive
分类号 A61K9/00;A61K31/53;A61K47/34;A61K47/10;A61K47/12;A61K47/26;A61K31/519;A61K31/4985 主分类号 A61K9/00
代理机构 代理人
主权项 1. A method of preventing or treating a sexual dysfunction, pulmonary hypertension, a vascular or cardiac or neurodegenerative condition, a physical injury, multiple sclerosis or fetal growth restriction in an individual, comprising delivering by sublingual administration as a spray a composition that comprises: a PDE5 inhibitor; and a carrier in which said PDE5 inhibitor is soluble or forms a suspension or emulsion.
地址 Norwich, Norfolk GB