发明名称 |
METHOD FOR PRODUCING PHENYL-SUBSTITUTED HETEROCYCLIC DERIVATIVE |
摘要 |
<p>The present invention is a method for producing a phenyl-substituted heterocyclic derivative represented by general formula (1), which has a step wherein a heteroaromatic compound represented by general formula (2) is reacted with a phenol derivative represented by general formula (3) in the presence of a nickel compound, 1,2-bis(dicyclohexylphosphino)ethane, and a base.</p> |
申请公布号 |
EP2774923(A4) |
申请公布日期 |
2014.12.31 |
申请号 |
EP20120845027 |
申请日期 |
2012.10.10 |
申请人 |
NATIONAL UNIVERSITY CORPORATION NAGOYA UNIVERSITY |
发明人 |
ITAMI, KENICHIRO;YAMAGUCHI, JUNICHIRO;MUTO, KEI |
分类号 |
C07D263/32;C07B61/00;C07D263/34;C07D263/56;C07D263/57;C07D277/22;C07D277/66;C07D413/04;C07D471/08 |
主分类号 |
C07D263/32 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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