发明名称 CYCLIC PYRIMIDIN-4-CARBOXAMIDES AS CCR2 RECEPTOR ANTAGONISTS FOR TREATMENT OF INFLAMMATION, ASTHMA AND COPD
摘要 The present invention relates to novel antagonists for CCR2 (CC chemokine receptor 2) and their use for providing medicaments for treating conditions and diseases, especially pulmonary diseases like asthma and COPD, of Formula (I), wherein A is selected from among a single bond, -CH-, -O-, -S-, and -NH-; wherein n is 1, 2 or 3; Z is C or N, the other variables are as defined in the claims, as well as in form of their acid addition salts with pharmacologically acceptable acids.
申请公布号 EA020548(B1) 申请公布日期 2014.12.30
申请号 EA20110000942 申请日期 2009.12.17
申请人 BOEHRINGER INGELHEIM INTERNATIONAL GMBH 发明人 EBEL HEINER;FRATTINI SARA;GIOVANNINI RICCARDO;HOENKE CHRISTOPH;TRIESELMANN THOMAS;TIELMANN PATRICK;SCHEUERER STEFAN;HOBBIE SILKE, (MARIE KATRIN);BUETTNER FRANK
分类号 C07D401/06;A61K31/506;A61P29/00;C07D401/14;C07D403/06;C07D407/14;C07D413/14;C07D471/10 主分类号 C07D401/06
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