发明名称 |
PROCESS FOR PREPARING PYRIDINONE COMPOUNDS |
摘要 |
<p>Disclosed herein is a process for preparing a compound of Formula (I), comprising the steps of: (a) reacting an aniline compound of Formula (II) and an carboxylic acid compound of Formula (III) or an activated carboxylic acid compound thereof, to provide a compound of Formula (IV); and (b) converting said protected amine group attached to said compound of Formula (IV) to an amine group to provide said compound of Formula (I); wherein PAm is a protected amine group. Processes to prepare the compounds of Formulae (II), (III), and (IV) are also disclosed.</p> |
申请公布号 |
EP2235001(B1) |
申请公布日期 |
2014.12.24 |
申请号 |
EP20090703743 |
申请日期 |
2009.01.22 |
申请人 |
BRISTOL-MYERS SQUIBB COMPANY |
发明人 |
LIVINGSTON, ROBERT C.;GALLAGHER, WILLIAM P. |
分类号 |
C07D401/12;A61K31/4427;A61P35/00;C07D213/63;C07D213/74 |
主分类号 |
C07D401/12 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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