发明名称 PROCESS FOR PREPARING PYRIDINONE COMPOUNDS
摘要 <p>Disclosed herein is a process for preparing a compound of Formula (I), comprising the steps of: (a) reacting an aniline compound of Formula (II) and an carboxylic acid compound of Formula (III) or an activated carboxylic acid compound thereof, to provide a compound of Formula (IV); and (b) converting said protected amine group attached to said compound of Formula (IV) to an amine group to provide said compound of Formula (I); wherein PAm is a protected amine group. Processes to prepare the compounds of Formulae (II), (III), and (IV) are also disclosed.</p>
申请公布号 EP2235001(B1) 申请公布日期 2014.12.24
申请号 EP20090703743 申请日期 2009.01.22
申请人 BRISTOL-MYERS SQUIBB COMPANY 发明人 LIVINGSTON, ROBERT C.;GALLAGHER, WILLIAM P.
分类号 C07D401/12;A61K31/4427;A61P35/00;C07D213/63;C07D213/74 主分类号 C07D401/12
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