发明名称 BENZYL PIPERIDINE COMPOUNDS AS LYSOPHOSPHATIDIC ACID (LPA) RECEPTOR ANTAGONIST
摘要 The invention provides novel substituted benzyl piperidine compounds according to Formula (I) as lysophosphatidic acid (LPA) receptor antagonists, their manufacture and use for the treatment of proliferative or inflammatory diseases, such as cancer, fibrosis or arthritis.
申请公布号 WO2013045028(A9) 申请公布日期 2014.12.24
申请号 WO2012EP03771 申请日期 2012.09.07
申请人 MERCK PATENT GMBH;SCHIEMANN, KAI;STAEHLE, WOLFGANG;BUSCH, MICHAEL;WIENKE, DIRK;POESCHKE, OLIVER;BURGER, CHRISTA 发明人 SCHIEMANN, KAI;STAEHLE, WOLFGANG;BUSCH, MICHAEL;WIENKE, DIRK;POESCHKE, OLIVER;BURGER, CHRISTA
分类号 C07D401/04;A61K31/4523;A61P29/00;A61P35/00;C07D407/04;C07D417/04 主分类号 C07D401/04
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