发明名称 PROCESS FOR CABAZITAXEL
摘要 The present invention provides an improved process for the preparation of 4α-acetoxy-2α-benzoyloxy-5&bgr;,20-epoxy-1&bgr;,13α-dihydroxy-7&bgr;,10&bgr;-dimethoxy-9-oxo-11-taxene (7&bgr;,10&bgr;-dimethoxy-10-deacetoxybaccatin III). The present invention also provides a novel process for the preparation of cabazitaxel.
申请公布号 WO2014199401(A2) 申请公布日期 2014.12.18
申请号 WO2014IN00395 申请日期 2014.06.12
申请人 HETERO RESEARCH FOUNDATION;PARTHASARADHI REDDY, BANDI;RATHNAKAR REDDY, KURA;MURALIDHARA REDDY, DASARI;VENKAT NARSIMHA REDDY, ADULLA;VAMSI KRISHNA, BANDI 发明人 PARTHASARADHI REDDY, BANDI;RATHNAKAR REDDY, KURA;MURALIDHARA REDDY, DASARI;VENKAT NARSIMHA REDDY, ADULLA;VAMSI KRISHNA, BANDI
分类号 C07D305/14 主分类号 C07D305/14
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